1、Hotline: 400-820-3792Inhibitors Agonists Screening Librarieswww.MedChemEDIM-C-pPhCO2MeCat. No.: HY-112056CAS No.: 151358-48-4分式: CHNO分量: 380.44作靶點: Others作通路: Others儲存式: Powder -20C 3 years4C 2 yearsIn solvent -80C 6 months-20C 1 month溶解性數(shù)據(jù)體外實驗 DMSO : 125 mg/mL (328.57 mM)* means soluble, but satura

2、tion unknown.Mass Solvent1 mg 5 mg 10 mg Concentration制備儲備液1 mM 2.6285 mL 13.1427 mL 26.2854 mL5 mM 0.5257 mL 2.6285 mL 5.2571 mL10 mM 0.2629 mL 1.3143 mL 2.6285 mL請根據(jù)產(chǎn)品在不同溶劑中的溶解度，選擇合適的溶劑配制儲備液，并請注意儲備液的保存式和期限。體內(nèi)實驗 請根據(jù)您的實驗動物和給藥式選擇適當?shù)娜芙獍?，配制前請先配制澄清的儲備液，再依次添加助溶?為保證實驗結(jié)果的可靠性，體內(nèi)實驗的作液，建議您現(xiàn)現(xiàn)配，當天使；澄清的儲備液可以根據(jù)儲

3、存條件，適當保存；以下溶劑前的百分 指該溶劑在您配制終溶液中的體積占)：1. 請依序添加每種溶劑： 10% DMSO 40% PEG300 5% Tween-80 45% salineSolubility: 2.08 mg/mL (5.47 mM); Clear solution2. 請依序添加每種溶劑： 10% DMSO 90% (20% SBE-CD in saline)Solubility: 2.08 mg/mL (5.47 mM); Clear solution1/2 Master of Small Molecules 您邊的抑制劑師www.MedChemEBIOLOGICAL ACT

4、IVITY物活性 DIM-C-pPhCO2Me是核受體 4A1 (NR4A1) 拮抗劑 1。具有抗腫瘤活性 1。IC50 & Target Nuclear receptor 4A1 (NR4A1) 1REFERENCES1. Hedrick E, et al. Nuclear Receptor 4A1 (NR4A1) as a Drug Target for Renal Cell Adenocarcinoma. PLoS One. 2015 Jun2;10(6):e0128308.McePdfHeightCaution: Product has not been fully validated for medical applications.For research use only.Tel: 400-820-3792;Fax: 021