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第1題Whichiswrongaboutthedescriptionofthedrug?()AAchemicalsubstanceB?AchemicalthatinterfereswithcellularmetabolicactivityCAsubstancethataffectsthephysiologicalfunctionsofthebodyDHasthenourishment,thenutrition,thehealthcare,therehabilitationfunctionmaterial第2題Pharmacologyisanimportantsubjectinmedicalteachingbecause()AThemechanismofactionofthedrugwaselucidatedBImprovethequalityofdrugs,improvetheefficacyofdrugsCItprovidesexperimentaldataandtheoreticalbasisforthedevelopmentofnewdrugsDItprovidesatheoreticalbasisforguidingrationaldruguseinclinicalpractice第3題Themethodofpharmacologyisexperimentalmeans()AStrictlycontroltheconditionandobservethelawandprincipleofdrugactiononthebodyBUsinganimalsforexperimentalresearchCThedrugwasstudiedinvitroandinvivoDTheexperimentaldataprovidedhaveimportantreferencevalueforclinic第4題Pharmacodynamicsisresearch()AClinicalefficacyofdrugsBWaystoimprovetheefficacyofdrugsCHowtoimprovedrugqualityDDrugactiononthebodyandthemechanismofaction第5題Pharmacokineticsisresearch()ADrugchangesinthebodyandtheirregularityBHowdodrugsaffectthebodyCArationalmedicationregimenDThedynamicchangesofdrugsandtheirlaws第6題Pharmacologyisresearch()ApharmacodynamicsB?pharmacokineticsCdrugDDrug-bodyinteractionanditslaw第7題Newdrugsmustbeprovided()forclinicaltrialsASystematicpharmacologicalresearchdataBAcuteandchronictoxicitywereobservedCLD50DPreclinicaldata第8題Theresearchobjectofpharmacologyis()AhumanbodyBbodyCAnimalpathologicalmodelDhealthyanimal第9題Theresearchobjectofexperimentalpharmacologyis()AanimalBbodyChumanbodyDhealthvolunteer第10題Theresearchobjectofclinicalpharmacologyis()AhumanbodyBbodyCAnimalpathologicalmodelDhealthvolunteerEorganism正確答案:E第1題Mostdrugsenterthebodybyoneofthefollowingmechanisms()AfaciliteddiffusionBsimplediffusionCactivetransportDfiltration第2題Activetransportischaracterizedby()ATransportbycarrier,noenergyisrequiredBThroughcarriertransport,energyisrequiredCNocarriertransport,noenergyconsumptionDWithoutcarriertransport,energyisrequired第3題Easydiffusionis
()ATransmembranetransportbycarrieragainstconcentrationgradientB()Nocarrier,trans-membranetransportalongconcentrationgradientCRelyingonthecarrier,trans-membranetransportalongtheconcentrationgradientDsimplediffusion第4題Whichofthefollowingstatementsaboutactivedrugtransportisfalse()AIttakesenergyBCanbedisturbedbyotherchemicalsCChemicalstructurespecificityDEquilibriumisreachedfasterthanpassivetransport第5題Whichofthefollowingstatementsaboutoraladministrationisfalse(
)AAfterabsorption,itenterstheliverviatheportalveinBAbsorptionisrapidandcompleteCThereisfirstpasseliminationDThesmallintestineisthemainsiteofabsorption第6題The
administrationrouteofthefirstpasselimination
is(
)
ArectaladministrationBsublingualadministrationCintravenousadministrationDoralmedication第7題Thedrugentersthebloodstream,first
(
)
AItACTSonthetargetorganBMetabolizeintheliverCExcretioninthekidneyDBindstoplasmaproteins第8題FluidpHaffectsdrugtransportanddistributionbecauseitaltersthedrug
(
)AwatersolubilityBlipidsolubilityCpKaDdegreeofdissociation第9題Adrugthatdoesnotdirectlycauseitseffectis
(
)
AAdrugthatismetabolizedbytheliverBAdrugthatbindstoaplasmaproteinCDrugsinthecirculationofbloodDMedicationsthatreachthebladder第10題Liverdrugenzymesarecharacterizedby
(
)
ALimitedactivity,highspecificity,largeindividualdifferencesBHighactivity,highspecificity,largeindividualdifferencesCHighactivity,highspecificity,smallindividualdifferencesDLimitedactivity,lowspecificity,largeindividualdifferencesChapter3test第1題Theintrinsicactivity()ofthedrugrefersto
()ATheabilityofdrugstopenetratebiofilmsBTheabilityofdrugstostimulatereceptorsCThewater-solublesizeofthedrugDTheaffinityofthedrugforthereceptor第2題Thedualityofdrugactionmeans
()ABoththerapeuticandsymptomatictreatmentBBothsideeffectsandtoxiceffectsCBoththerapeuticeffectsandadversereactionsDHasbothlocalandsystemiceffects第3題Takingbarbituratesappearsina"hangover"phenomenon,called
()AAftermathBReboundphenomenonCspecificheterogeneousreactionDAllergicreactions第4題Theallergicreactionproducedbythedrugdependson(
)
APharmacodynamicproperties
BPharmacokineticpropertiesCBothAandB
DNonAnonB第5題Thecharacteristicsofcompetitiveantagonistsare
()AAffinitytothereceptorandintrinsicactivityBHaveaffinityforthereceptor,butnointrinsic
activityCNoaffinityforreceptors,butintrinsicactivityDNoaffinityforreceptors,nointrinsicactivity第6題Thefollowingstatementisnotcorrect()AConcentration-effectrelationshipismorecommonlyusedinpharmacologicalresearchBThepharmacologicaleffectisexpressedinapositiveornegative,allornothingway,calledqualitativereactionCThesafetyindexindicatedbyLD5/ED95isrelativelyreliableDTherelativeconcentrationordosethatcancauseanequivalentresponse(generallyusing50%effectamount)iscalledpotency第7題Theeffectofintramuscularinjectionofatropinetotreatbiliarycolicandcauseblurredvisioniscalled()AToxicityBSideeffectsCEfficacyDAllergy第8題Thetoxicreactionofthedrugis()AAnallergicreactionBReactionsunrelatedtothepurposeoftreatmentwhenusingtherapeuticdosageCDamagetothebodyduetoexcessivedosageorthebodyisparticularlysensitivetothedrugDAspecificreactioncausedbyanabnormalgeneticbiochemicalmechanism第9題Theselectivityofthedrugdependson(
)C.
BothAPharmacodynamicpropertiesBPharmacokineticproperties
CBothAandBDNonAnonB第10題Thedecreaseinsensitivitycausedbycontinuousmedicationiscalled()ADrugresistanceBToleranceCHighsensitivityDDependenceChapter4test第1題Cholinergicnervedoesnotinclude
()AAllpresympatheticfibersBMostpost-sympatheticfibersCAllparasympatheticpreganglionicfibersDPost-sympatheticfibersinnervatingthesweatglands第2題Whichofthefollowingaminoacidsistherawmaterialforsynthesisofnorepinephrine()AmethionineBglutamicacidCtyrosineDlysine第3題Themaineliminationmethodofnorepinephrineis()ADestroyedbycatecholoxygenmethyltransferaseBReuptakebynerveendingsCDestroyedbyacetylcholinesteraseDDamagedbyphenylethylaminenitrogenmethyltransferase第4題Themainwaytoeliminateacetylcholineis()AHydrolyzedbymonoamineoxidaseBHydrolyzedbyphosphodiesteraseCHydrolyzedbyacetylcholinesteraseDHydrolyzedbycholineacetylase第5題Thetransmitterreleasedbythefibersaftertheparasympatheticgangliais()ASuccinylcholineBMethacholineCNicotineDAcetylcholine第6題TheenzymethatinactivatesNAisCatecholaminemethyloxytransferase()第7題Norepinephrinenerveexcitementcannotenhancecardiaccontractility()第8題Cholinergicnerveexcitementcancauseskeletalmusclerelaxation()第9題MreceptorblockcancauseDilatedpupilsandIncreasedheartrate()第10題βreceptoractivationdecreasedheartrate()Chapter5test第1題muscariniccholinoceptoragonistsmaycausevasodilationthroughthereleaseofendothelial()AHistamineBNorepinephrineCacetylcholineDNitricoxide第2題Apatientwithanacuteattackofglaucomaistreatedwithpilocarpine.Theprimaryreasonforitseffectivenessinthisconditionisits:()AactiontoterminateacetylcholinesteraseBslectivelyfornicotinicreceptorsCabilitytoinhibitsecretions,suchastears,salivaandsweatDabilitytolowerintraocularpressure第3題apatientwithmyastheniagraviswouldbetreatedwith()AdonepezilBedrophoniumCatropineDneostigmine第4題whichclassofmedicationsdoesbethanecholbelongto?()AnicotinicblockersBalpha-agonistsCbeta1-blockersDmuscarinicreceptors第5題Whichofthefollowing
agentsdoesnotbindtomuscrinicreceptordirectly?()ApilocarpineBcarbacolCneostigmineDatropine第6題Whichofthefollowingtheagentscouldnotbeusedforpateintswithalzhemierdisease?()AneostigmineBtacrineCDonepezilDgalanthamine第7題Nicotineinlowdosesmaycause(
)ADecreasedtoneandmotoractivityofthesmallintestineBStimulationoftherespiratoryraleanddepthCMiosisDBradycardia第8題whichofthefollowingpharmacologicaleffectsof
neostigmine
isthestrongest?()AskeletalmuscleconstrictionBstimulatesmovementofgastrointestinalsmoothmuscleCincreaseglandularsecretionDinhibitioncardiacfunction第9題Neostigminewilleffectivelyantagonizeskeletalmusclerelaxationproducedby()ANicotineBSuccinylcholineCDiazepamDBaclofen第10題Thecholinesteraseinhibitorthatisusedinthediagnosisofmyastheniagravisis()AEdrophoniumchlorideBAmbenoniumchlorideCPhysostigminesalicyhteDPyridostigminebromideChapter6test第1題WhichOfthefollowing,whichwillnotbeblockedbyatropineandscopolamine?()ABradycardiaBSalivarysecretionCBronchoconstrictionDSkeletalmusclecontraction第2題Whichofthefollowingantimuscarinicdrugsisusedbyinhalationinthetreatmentofbronchialasthma?()ADicyclominehydrochlorideBCyclopentolatehydrochlorideCIpratropiumbromideDMethscopolaminebromide第3題Whichofthefollowingisnottheeffectofatropine?()AInhibitsglandsecretionBRelaxessmoothmuscleCIncreasesintraocularpressureDincreasesbloodpressure第4題Whichofthefollowingcouldbeusedinparkinsondisease?()AatropineBAnisodamineCScopolamineDpirenzepine第5題Allofthefollowingagentscouldbeused
topreventasphyxia-inducedbygeneralanesthesia
,(
)is
thebestselection.AatropineBScopolamineCdiazepamDNeostigmine第6題WhichofthefollowingagentsisselectiveMuscrinicreceptorantagonist?()AAtropineBScopolamineCTelenzepineDBenactyzine第7題Neostigminewilleffectivelyantagonizeskeletalmusclerelaxationproducedby()APancuroniumBSuccinylcholineCDiazepamDNicotine第8題Whichofthefollowingstatementsiscorrectaboutitseffectoneyes?()Amydriasis,increaseintraocularpressure,
spasmofaccommodationBmydriasis,increaseintraocularpressure,
paralysisofaccommodationCmyosis,decreaseintraocularpressure,
paralysisofaccommodationDmyosis,
decreaseintraocularpressure,
spasmofaccommodation第9題WhichofthefollowingagentsisbestforVisceralcolic?()AatropineBsocoplamineCAnisodamineDpirenzepine第10題Atropineatlargedosemaycausethe
toxicity,whichofthefollowingagentscanrelievethetoxicity?()ApilocarpineBnicotineCdiazepamDneostigmineChapter7test第1題Whichoffollowingdrugcanincreasethebloodflowofrenal?()AAdrenalineBIsoproterenolCEphedrineDDopamine第2題Thefirstchoiceofencounteringpenicillin-inducedanaphylacticshockis()ANorepinephrineBIsoproterenolCAdrenalineDDopamine第3題Whenshockiscomplicatedbyacuterenalfailure,itisbesttochoose()ADopamineBMetaraminolCAdrenalineDDobutamine第4題()canselectivelyactive
β1receptorADopamineBDobutamineCAdrenalineDEphedrine第5題whichoffollowingadrenalinedrughasanexcitatoryeffectonthecenterandcanpromotethereleaseofnerveendingtransmitters?()AAdrenalineBIsoproterenolCDopamineDEphedrine第6題()cantreatnasalmucosacongestioncausedstuffynose.ANorepinephrineBAdrenalineCIsoproterenolDEphedrine第7題whichofthefollowingdiseaseisnotcontraindicationtoadrenaline?()ABronchialasthmaBHyperthyroidismCDiabetesDCardiogenicasthma第8題whichisthemainrouteofremovingnorepinephrine()AOxidatedbymonoamineoxidaseBMetabolizedbycatecholO-methyltransferaseCRecapturedbypresynapticmembraneDReingestedbytheliver第9題ThepharmacologicaleffectsofIsoproterenolare()AStimulationoftheheart,increaseinsystolicanddiastolicbloodpressure,relaxbronchialsmoothmuscle,
loosenbronchialsmoothmuscleBStimulationoftheheart,increaseinsystolicbloodpressure,decreaseindiastolicbloodpressure,loosenbronchialsmoothmuscleCStimulationoftheheart,decreaseinsystolicanddiastolicbloodpressure,loosenbronchialsmoothmuscleDStimulationoftheheart,increaseinsystolicanddiastolicbloodpressure,contractionofbronchialsmoothmuscle第10題whichoffollowingadrenalinedrughasanexcitatoryeffectonthecenterandcanpromotethereleaseofnerveendingtransmitters?()ANotinfluencedBStrengthenCReversedDWeakenChapter8test第1題Whichofthefollowingdrugcanbeusedtotreatperipheralvasospasmdiseases?()AScopolamineBPhentolamineCAdrenalineDPropranolol第2題()caninducetheacuteattackofbronchialasthmaAPhenoxybenzamineBAdrenalineCPhentolamineDPropranolol第3題Thesystemicbloodpressureresponsestoepinephrinewillbereversedbyusing()AD1receptorblockerBMreceptorblockerCβreceptorblockerDαreceptorantagonist第4題()canselectivelyblock
α1receptorAClonidineBPrazosinCPhentolamineDTolazoline第5題Thefollowingoptionsarethepharmacologicaleffectsofpropranololexcept()AContractilebronchialsmoothmuscleBReducemyocardialcontractilityCConstrictbloodvesselsDReducemyocardialoxygenconsumption第6題Whichoffollowingoptionisnottheindicationofphentolamine?()APeripheralvasospasmdiseaseBPreoperativeapplicationofpheochromocytomaCCoronaryheartdiseaseDSepticshock第7題Whichofthefollowingisnotacontraindicationforpropranolol?()AVentriculararrhythmiaBCardiogenicshockCBronchialAsthmaDHypotension第8題()isnon-selective
β
receptorblockerwithoutinherentsympathomimeticactivityAMetaprololBAtenololCLabetalolDPropranolol第9題Atenololandpropranololaredifferentin()ANoinherentsympathomimeticactivityBUsewithcautioninasthmapatientsCTreatmentofhypertensionDSelective
β1receptorantagonist第10題Whichoneoffollowingβ-blockerhastheeffectonreducingintraocularpressure?()ATimololBPropranololCAtenololDMetaprololChapter9test第1題Thereasonwhycabidobaisinco-operationwithlevodobais()AIncreasedopamineconcentrationinthebrainandenhanceefficacyBSlowingl-dobakidneyexcretionandenhancingefficacyCDirectlyexciteddopaminereceptorstoenhanceefficacyDInhibitingdopaminere-intaketoenhancethecentralefficacyofl-dopa第2題WhatkindsofdrugscurrentlytreatParkinson'sdiseaseis
()AAdrenalinedrugsBDopaminedrugsCAntihistaminesDAnticholinergase第3題levodopais
()AInhibitionofperipheralaminoaciddeoxidaseBExcitedcentraldopaminereceptorCConversiontodopamineinthecenterDBlockingcentralcholinereceptors第4題Cabidopawill()AInhibitionofperipheraldopadecarboxylaseBExcitedcentraldopaminereceptorCConversiontodopamineinthecenterDBlockingcentralcholinereceptors第5題Bromocriptinewill()AInhibitionofperipheralaminoaciddeoxidaseBExcitedcentraldopaminereceptorCConversiontodopamineinthecenterDBlockingcentralcholinereceptors第6題VitaminB6inmultivitaminpreparationscanreducetheeffectoflevodopa()第7題Thecombinationofl-dopaandmonoamineoxidaseinhibitorscancausehypertension()第8題leprodopa
isavailablewhenParkinson'ssyndromethatoccursinthetreatmentofschizophreniawithchlopromazin()第9題?Levodobausetogetherwithadrenalinecaninducearrhythmia()第10題L-dobacanbeuseddopaminetogetherwithtotreatParkinson'sdisease()Chapter10test第1題Thefollowingdescriptionofbenzodiazepam,whichoneisnotcorrect()AEnhancegabA'sneurotransmitterfunctionBCanbeusedasapre-anaestheticadministration.CLong-termnon-addictiveDrelaxantofcentralbonemusclepine第2題Themechanismofcentralinhibitionofbenzodiazepine
is()ADirectlyactingonthegamma-aminobutyricacid(GABA)receptor,openingtheCl-channelBDirecteffectonbenzodiazepinereceptor,makingCl-channelopenCDirectlyactingonbenzodiazepinereceptors,promotingCL-channelopeningcausedbyGABADDirectlyactingonGABAreceptors,promotingCl-channelopeningduetobenzodiazepinereceptors第3題Themainreasonfortheclinicalreplacementofthetraditionalsedativehypnoticdrugofthebenzodiazepineclassis()ATheeffectofbenzodiazepineonfastwavesleeptimeisgreatBBenzodiazepinescancauseanesthesiaCSmalldosesofbenzodiazepinescanproducehypnoticeffectsDBenzodiazepineshavebetteranti-anxietyandcalmingeffects,goodsafety第4題EnhancedGABAinhibitionisduetotheincreaseinthefrequencyofCl-channelopeningdrugsis()ABenzodiazepinesBBarbitratesCSodiumPhentotoinDcabamazepine第5題Thenarrativeerroroftheadversereactionofbenzodiazepinesis()AOverdoseacutepoisoningcancausecomaandrespiratorysuppressionBLargescopeofsafety,fewerseriousconsequencesCIntravenouscardiovascularinhibitionDLong-termservicecanproducedependencebutisnotaddictive第6題Whenacutepoisoningofphenylbarbital,inordertospeedupitsexcretionfromthekidneys,themeasurestobetakenissodiumbicarbonatesolution()第7題Thedrugwhichhaslargesafetyrange,breathsuppressionintheeventofanoverdoseofacutepoisoningisdiazepam()第8題diazepamhastheeffectofantidepression.()第9題Inthecaseofacutepoisoningofbenzodiazepines,naloxonecanbeused.()第10題Theprocesscharacteristicsofbenzodiazepinesisgoodabsorptionoforalandmuscleadministration()Chapter11test第1題Chlorpromazinecannotbeusedforvomitingcausedby
()AUremiaBCancer?C.RadiationsicknessCMotionsickness第2題Whichisthebestanswertotheeffectofchlorpromazineonthereceptor()ABlockDA,α,MreceptorsBBlockdopaminereceptors,blockalphareceptorsCBlockdopaminereceptors,blockMreceptorsD
Blockαreceptor,blockMreceptor第3題Misrepresentationoftheantipsychoticeffectofchlorpromazine
()AHasastrongneurolepticeffectBCanquicklycontrolthepatient'sagitatedsymptomsCIneffectivefordepression,evenworseDGoodcurativeeffectonacuteschizophrenia,withradicaleffect第4題Thewrongstatementabouttheanpyreticeffectofchlorpromazineis()ANeedtocombinepethidineandpromethazineBInhibitionofbodytemperatureregulationcenterCNoeffectonnormalbodytemperatureDCanreducefeverbodytemperature第5題Lithiumcarbonateismainlyusedfortreatment()AAnxietyBSchizophreniaCManiaDParkinson'ssyndrome第6題Parkinson'ssyndromeisnotbelongtoExtrapyramidalreactionscausedbychlorpromazine()第7題Antipsychoticeffect:ChlorpromazineblocksD2receptorsinthemidbrain-limblobeandmidbrain-cortexpathways
()第8題Chlorpromazineblocksthesubstantianigra-striatalpathwayD2receptorcancause
extrapyramidalresponse()第9題ChlorpromazineblocksMcholinereceptorscancause
Drymouth,constipation,blurredvision()第10題ChlorpromazineblockstheD2receptorofCTZ
willcauseFailuretoregulatebodytemperature()Chapter12test第1題Themosteffectivetreatmentforsmallseizuresandineffectiveforothertypesofepilepsyisethosuximide()第2題Grand-malseizuresarenotpartoftheclinicaluseofphenytoin()第3題Thefirstchoiceformajorseizuresorpsychomotorseizuresiscarbamazepine()4.Thefirstchoiceformajorseizuresorpsychomotorseizuresiscarbamazepine(√)5.Thepreferreddrugforstatusepilepticusisdiazepam(√)第4題Phenytoinsodiumisadrugusedtotreatabsentseizures()第5題Ataxia,nystagmusisnotanadversereactionoflong-termuseofphenytoin()第6題Carbamazepine,phenytoinandsodiumvalproateareeffectiveforgrand-malseizureinepilepsy()第7題Themainclinicaluseofcarbamazepinedoesnotincludebradyarrhythmia()第8題Drugswithgoodefficacyformajorseizuresorlocalizedseizuresarephenytoinandcarbamazepine()Chapter13test第1題MorphinecanbeusedforBronchialasthma()第2題Morphineacutepoisoningcanchoose
Atropinetorescue()第3題Comparedwithmorphine,pethidineismorecommonlyusedmainlyduetostrongerrespiratorydepression()第4題Thereasonwhypethidineisnotusedalonetotreatbiliarycolicdueto
itcancausebiliarysphincterspasm()第5題Theanalgesiceffectofmorphineismostsuitableforthediagnosisofunexplainedacuteabdominalpain()第6題ForBilecolic,atropine+pethidine
is
bestused()第7題Morphinehasstrongeranalgesiceffectthandulending()第8題Morphineismoreaddictivethandulending()第9題Pethedineandmorphinebothhavestrongantitussiveeffects()第10題Women'sdeliveryisnotacontraindicationformorphine()Chapter14test第1題Themainsiteandmechanismofaspirin'sanalgesiceffectisthesynthesisofPGwhenpreventinginflammationintheperiphery()第2題Thedrugwithoutanti-inflammatoryandanti-rheumaticeffectisacetaminophen()第3題AspirinpreventsthrombosisbyinhibitingcyclooxygenaseactivityandreducingTXA2productioninplatelets()第4題Aspirinsalicylicacidreactioncanberescuedwithpotassiumchloride()第5題Theprincipleofaspirin'santipyreticeffectistoinhibitprostaglandinsynthesis()第6題Gastrointestinalreactionisacommonadversereactionforaspirin()第7題Aspiriniseffectiveagainstbacterialinflammation()第8題Excessiveacetaminophencancauselivernecrosis()第9題Commonadversereactionsofaspirinincludegastrointestinalreactionsandarrhythmias()第10題Aspiriniscontraindicatedinbronchialasthma()Chapter15test第1題Theprincipleofcardiactoxicitycausedbycardiacglycosideis
()AincreaseK+Bincardiomyocytes,increaseCa2+incardiomyocytesC.ExciteNa+-K+-ATPaseofmyocardialcellmembraneCInhibitNa+-K+-ATPaseofmyocardialcellmembrane第2題Captoprilwillleadto()AElevatedbloodpotassiumBGumhyperplasiaCAnaphylacticshockDReflexheartraterise第3題Thecommoneffectofnitroglycerin,β-blockerandcalciumantagonistonanginapectorisis()ADilatebloodvesselsBInhibitmyocardialcontractilityCReducemyocardialoxygenconsumptionDSlowdownheartrate第4題Whichofthefollowingadversereactionsisnotrelatedtotheroleofnitroglycerinindilatingbloodvessels()AIncreasedheartrateBOrthostatichypotensionCElevatedintraocularpressureDMeteorhemoglobinemia第5題Itisbesttochooseatrioventricularblockorsinusbradycardiacausedbycardiacglycosidepoisoning()AaminophyllineBphenytoinCatropineDisoproterenol第6題Thedrugthatexertsantihypertensiveeffectbyinhibitingangiotensinconvertingenzymeis()AClonidineBEnalapril(PhenylProline)CReserpineDSodiumnitroprusside第7題Captoprilcombinedwithpotassium-retainingdiuretics,itiseasytocausehyperkalemia
()第8題Forpatientswithstableangina,youshouldchoosenitroglycerin.
()第9題WhendigoxinisusedforCHFtreatment,itcanreducebloodvolumeandreduceheartload
.()第10題Betablockerscanincreasemyocardialcontractilityandincreasecardiacoutputtogivetreatmentforheartfailure.()Chapter16test第1題Whichmedicinedoesnotincreasetheheartratewhendilatingbloodvesselstolowerbloodpressure()AHydralazineBPhentolamineCNitroglycerinDLabello第2題Forhypertensionwithpepticulcers,thepreferredantihypertensivedrugis()APrazosinBMethyldopaCNifedipineDClonidine第3題AngiotensinⅠconvertingenzymeinhibitoris()ASodiumnitroprussideBCaptopriCHydralazinePyridazineDPrazosin第4題Thedrugthatreducesbloodpressurebydirectlyblockingtheα1receptoris()ARisapingBMethyldopaCPrazosinDNifedipine第5題Thecentralantihypertensivedrugis()AClonidineBRisapingCLabellolDHydralazine第6題Thedrugthatexertsanantihypertensiveeffectbyblockingα1andβreceptorsis()APrazosinBPropranololCNifedipineDLabello第7題Themedicinethatlowersbloodpressurebyaffectingtherenin-angiotensin-aldosteronesystemis()ARisapingBPrazosinCMethyldopaDCaptopril第8題Whichdrugshouldnotbeusedforhypertensionwithheartfailure()APropranololBCaptoprilCPrazosinDHydrochlorothiazide第9題Thestrongestantihypertensiveeffectis()Aα-MethyldopaBClonidineCGuanfasinDMoxonidine第10題Whichofthefollowingantihypertensivedrugsislikelytocausethe"firstdosephenomenon"()AHydrochlorothiazideBCaptoprilCPrazosinDPropranololChapter17test第1題Whichofthefollowingcardiacglycosidesismostcompletelyabsorbedafteroraladministration?()AdigitalisglycosideBdigoxinCflavosideDgeninC第2題Whichofthefollowingdrugscanincreasethebloodconcentrationofdigoxin
?()AKClBspironolactoneCcholestyramineDquinidine第3題Themostcommonearlysymptomofcardiacglycosidepoisoningis?()AECGhasashortenedQ-TintervalBheadacheCgastrointestinalreactionDatrioventricularblock第4題Sinusbradycardiacausedbycardiacglycosidepoisoningcanbeused()ApotassiumchlorideBAtropineCLidocaineDEpinephrine第5題Thefollowingdrugsarenotsuitableforthetreatmentofheartfailure?()AAdrenalineBNitroglycerinCHydrochlorothiazideDPrazosin第6題Theprincipleofcardiactoxicitycausedbycardiacglycosideis()AInhibitNa+-K+-ATPaseofmyocardialcellmembraneBExciteNa+-K+-ATPaseofmyocardialcellmembraneCIncreaseK+incardiomyocytesDIncreaseCa2+incardiomyocytes第7題Whichofthefollowingdrugsisbannedfromcardiogenicasthma()AMorphineBsildilanCEpinephrineDAminophylline第8題Thereasonwhycardiacglycosideslowstheventricularrateinpatientswithatrialfibrillationis()?ADecreasetheautonomyofatrialmusclesBDecreasetheautonomyofventricularmusclesCImprovemyocardialischemiaDIncreasetheoccultconductionintheatrioventricularnode第9題Cardiacglycosideisbetterforheartfailurecausedbywhichofthefollowingdiseases()AhighbloodpressureBsevereanemiaCHyperthyroidismDVB1deficiency第10題Cardiacglycosidesareprohibitusedin
()AHeartfailurecausedbyhypertensionBAtrialfibrillationCsupraventriculartachycardiaDventriculartachycardiaChapter18test第1題Whichofthefollowinganti-arrhythmiasagentscan
blockcaciumchannel?()AverapamilBprocaineClidocaineDquinidineEflecainide第2題Whichofthefollowingagentscanbeusedinventriculartachyarrhythmiacausedbyacutemyocardialinfarction.()ALidocaineBquinidineCpropranololDverapamilEamiodarone第3題suppressionofarrhythmiasresultingfromareentryfocusismostlikelytooccurifthedrug()
AhasvagomimeticeffectsotheAVnodeBisabeta-blockerCconvertsaunidirectionalblocktoabidrectionalblockDslowsconductionthroughtheatriaEhasatropine-likeeffectsontheAVnode第4題whichofthefollowingeffectsofdrugsfortachyarrhythmiasisnotcorrect.()AreductionofautomaticityBslowingdownconductionofatrialventricularnodeconductionCeliminationofreentryDprolongationofERPandAPDEaccelerationofautodepolarizationofpacemakers正確答案:E第5題Howdoesdigoxinworkinatrialfibrillation?()AitdecreasesintracellularsodiumandincreasesintracellularpotassiumBitlowersintracellularcalciumCitdecreasesstrokevolumeandcardiacoutputDitdiminsheseliminationofsodiumandwaterEitincreasesvagalactivityanddecreas
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